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TGX221

Synonyms

SourcesNames Used
GDSC1000TGX221
CTRPv2TGX-221
PharmacoGx TGX221

External IDs

DatabaseIdentifier
Smiles: CC1=CN2C(=O)C=C(N=C2C(=C1)C(C)NC3=CC=CC=C3)N4CCOCC4
Inchikey: CPRAGQJXBLMUEL-UHFFFAOYSA-N
Pubchem: 9907093

Annotated Targets

PIK3CB, PIK3CD

FDA Approval Status

Not Approved
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Top molecular features associated with response to TGX221


Feature TypeStandardized
Nominal ANOVA
mRNA BDH2 CTRPv2 pan-cancer AAC 0.19 7e-07
mRNA SP110 CTRPv2 pan-cancer AAC 0.19 8e-07
mRNA SLC16A4 GDSC1000 pan-cancer AAC 0.27 9e-07
mRNA CHST3 GDSC1000 pan-cancer AAC 0.26 1e-06
mRNA COL5A1 GDSC1000 pan-cancer AAC 0.3 1e-06
mRNA SYNPO CTRPv2 pan-cancer AAC 0.2 1e-06
mRNA COL5A2 GDSC1000 pan-cancer AAC 0.29 1e-06
mRNA TNFRSF13C CTRPv2 pan-cancer AAC 0.19 1e-06
mRNA TGFB2 CTRPv2 pan-cancer AAC 0.19 1e-06
mRNA NNMT GDSC1000 pan-cancer AAC 0.3 1e-06
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