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TGX221

Synonyms

SourcesNames Used
GDSC1000TGX221
CTRPv2TGX-221
PharmacoGx TGX221

External IDs

DatabaseIdentifier
Smiles: CC1=CN2C(=O)C=C(N=C2C(=C1)C(C)NC3=CC=CC=C3)N4CCOCC4
Inchikey: CPRAGQJXBLMUEL-UHFFFAOYSA-N
Pubchem: 9907093

Annotated Targets

PIK3CB, PIK3CD

FDA Approval Status

Not Approved
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Top molecular features associated with response to TGX221


Feature TypeStandardized
Nominal ANOVA
mRNA DPH6 GDSC1000 pan-cancer AAC -0.12 0.01
mRNA PYCR2 CTRPv2 pan-cancer AAC -0.11 0.01
mRNA COL7A1 GDSC1000 pan-cancer AAC 0.15 0.01
mRNA ICA1L CTRPv2 pan-cancer AAC -0.095 0.01
mRNA TSNARE1 CTRPv2 pan-cancer AAC -0.096 0.01
mRNA ALOX5AP CTRPv2 pan-cancer AAC 0.1 0.01
mRNA PPIC GDSC1000 pan-cancer AAC 0.17 0.01
mRNA PPIC CTRPv2 pan-cancer AAC 0.11 0.01
mRNA RP5-966M1.6 CTRPv2 pan-cancer AAC 0.099 0.01
mRNA TMEM263 GDSC1000 pan-cancer AAC 0.12 0.01
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