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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA ASB16 CTRPv2 pan-cancer AAC 0.23 2e-10
mRNA CASP10 CTRPv2 pan-cancer AAC 0.24 4e-10
mRNA CORO7 CTRPv2 pan-cancer AAC 0.27 4e-10
mRNA TXNDC11 CTRPv2 pan-cancer AAC 0.22 5e-10
mRNA B4GALT3 CTRPv2 pan-cancer AAC 0.21 5e-10
mRNA BCOR CTRPv2 pan-cancer AAC 0.23 5e-10
mRNA CLN6 CTRPv2 pan-cancer AAC 0.21 6e-10
mRNA SPCS1 CTRPv2 pan-cancer AAC 0.21 6e-10
mRNA SLC38A5 CTRPv2 pan-cancer AAC 0.23 7e-10
mRNA SNAP23 CTRPv2 pan-cancer AAC -0.22 8e-10
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