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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA RP4-583P15.14 CTRPv2 pan-cancer AAC 0.32 1e-20
mRNA LIME1 CTRPv2 pan-cancer AAC 0.31 7e-19
mRNA IGF1R GDSC1000 pan-cancer AAC 0.3 2e-17
mRNA PRDM1 CTRPv2 pan-cancer AAC 0.29 2e-16
mRNA TXNDC5 CTRPv2 pan-cancer AAC 0.27 5e-15
mRNA ZC2HC1B CTRPv2 pan-cancer AAC 0.26 1e-14
mRNA BLOC1S5-TXNDC5 CTRPv2 pan-cancer AAC 0.26 2e-14
mRNA INPP4A CTRPv2 pan-cancer AAC 0.27 2e-14
mRNA ITM2C CTRPv2 pan-cancer AAC 0.26 4e-14
mRNA RP4-583P15.15 CTRPv2 pan-cancer AAC 0.26 6e-14
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