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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA HDAC5 CTRPv2 pan-cancer AAC 0.26 1e-11
mRNA IL6R CTRPv2 pan-cancer AAC 0.24 3e-11
mRNA MYOM2 CTRPv2 pan-cancer AAC 0.24 4e-11
mRNA HPDL CTRPv2 pan-cancer AAC 0.24 4e-11
mRNA ITGB7 CTRPv2 pan-cancer AAC 0.22 5e-11
mRNA PMVK CTRPv2 pan-cancer AAC 0.24 6e-11
mRNA SWAP70 CTRPv2 pan-cancer AAC -0.22 7e-11
mRNA GPRIN3 CTRPv2 pan-cancer AAC 0.22 1e-10
mRNA DCC CTRPv2 pan-cancer AAC 0.22 1e-10
mRNA FOXO3 CTRPv2 pan-cancer AAC 0.22 2e-10
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