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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA PCLO GDSC1000 pan-cancer AAC -0.16 2e-06
mRNA PMF1 CTRPv2 pan-cancer AAC 0.17 2e-06
mRNA CD40 CTRPv2 pan-cancer AAC -0.16 2e-06
mRNA SLC25A20 CTRPv2 pan-cancer AAC 0.17 2e-06
mRNA BCL9 CTRPv2 pan-cancer AAC 0.17 2e-06
mRNA FKBP11 CTRPv2 pan-cancer AAC 0.16 2e-06
mRNA PTP4A3 CTRPv2 pan-cancer AAC 0.16 3e-06
mRNA ZNF740 GDSC1000 pan-cancer AAC 0.16 3e-06
mRNA ACTR2 CTRPv2 pan-cancer AAC -0.17 3e-06
mRNA TAF13 CTRPv2 pan-cancer AAC -0.18 3e-06
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