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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA IDH2 CTRPv2 pan-cancer AAC 0.12 0.002
mRNA SH3YL1 GDSC1000 pan-cancer AAC 0.12 0.002
mRNA CDH2 GDSC1000 pan-cancer AAC -0.13 0.002
mRNA WIPF1 CTRPv2 pan-cancer AAC -0.15 0.002
mRNA OR10H3 GDSC1000 pan-cancer AAC -0.1 0.002
mRNA FKBP1A CTRPv2 pan-cancer AAC -0.12 0.002
mRNA MBD3L4 CTRPv2 pan-cancer AAC 0.12 0.002
mRNA OR1Q1 CTRPv2 pan-cancer AAC 0.1 0.002
mRNA U2AF2 GDSC1000 pan-cancer AAC 0.11 0.002
mRNA SAMD4A CTRPv2 pan-cancer AAC -0.11 0.002
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