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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA NPIPA8 CTRPv2 pan-cancer AAC 0.12 0.001
mRNA POLR2M GDSC1000 pan-cancer AAC 0.11 0.001
mRNA PLEK CTRPv2 pan-cancer AAC -0.13 0.001
mRNA TFF1 FIMM pan-cancer AAC 0.49 0.001
mRNA ZFP36L1 CTRPv2 pan-cancer AAC -0.12 0.001
mRNA ZSCAN21 GDSC1000 pan-cancer AAC -0.11 0.001
mRNA PAX7 CTRPv2 pan-cancer AAC 0.12 0.001
mRNA PRSS3 CTRPv2 pan-cancer AAC 0.12 0.001
mRNA PFN1 CTRPv2 pan-cancer AAC -0.11 0.001
mRNA PGM3 CTRPv2 pan-cancer AAC -0.12 0.001
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