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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA TSHR CTRPv2 pan-cancer AAC 0.19 5e-08
mRNA SMAP2 GDSC1000 pan-cancer AAC -0.24 6e-08
mRNA DACH1 CTRPv2 pan-cancer AAC 0.19 6e-08
mRNA APH1A CTRPv2 pan-cancer AAC 0.18 6e-08
mRNA AMPD1 GDSC1000 pan-cancer AAC 0.18 6e-08
mRNA HNRNPK GDSC1000 pan-cancer AAC 0.18 7e-08
mRNA IRS2 GDSC1000 pan-cancer AAC 0.19 7e-08
mRNA SECISBP2 CTRPv2 pan-cancer AAC 0.2 8e-08
mRNA MAP4K2 CTRPv2 pan-cancer AAC -0.2 8e-08
mRNA MANEA CTRPv2 pan-cancer AAC 0.19 8e-08
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