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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA ABCD2 CTRPv2 pan-cancer AAC 0.2 1e-08
mRNA COQ8A CTRPv2 pan-cancer AAC 0.22 2e-08
mRNA PMF1-BGLAP CTRPv2 pan-cancer AAC 0.2 2e-08
mRNA DGAT2 CTRPv2 pan-cancer AAC 0.19 2e-08
mRNA CLK2 CTRPv2 pan-cancer AAC 0.22 2e-08
mRNA P2RX1 GDSC1000 pan-cancer AAC 0.22 3e-08
mRNA FAM19A5 CTRPv2 pan-cancer AAC 0.22 3e-08
mRNA PLD6 CTRPv2 pan-cancer AAC 0.2 3e-08
mRNA BHLHA15 CTRPv2 pan-cancer AAC 0.19 5e-08
mRNA ABHD14A CTRPv2 pan-cancer AAC 0.2 5e-08
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