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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA AMFR CTRPv2 pan-cancer AAC -0.17 4e-07
mRNA SP1 GDSC1000 pan-cancer AAC 0.17 4e-07
mRNA H1FX CTRPv2 pan-cancer AAC 0.18 5e-07
mRNA TADA1 CTRPv2 pan-cancer AAC 0.2 5e-07
mRNA PLEKHH3 CTRPv2 pan-cancer AAC 0.17 5e-07
mRNA ARMC2 CTRPv2 pan-cancer AAC 0.17 5e-07
mRNA WSCD1 CTRPv2 pan-cancer AAC 0.18 5e-07
mRNA RRAS2 CTRPv2 pan-cancer AAC -0.19 5e-07
mRNA UBE2J1 CTRPv2 pan-cancer AAC 0.19 5e-07
mRNA RTN4IP1 CTRPv2 pan-cancer AAC -0.17 6e-07
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