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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA IRF4 CTRPv2 pan-cancer AAC 0.2 9e-08
mRNA ACTR3 CTRPv2 pan-cancer AAC -0.19 9e-08
mRNA ST8SIA2 CTRPv2 pan-cancer AAC 0.22 9e-08
mRNA CDON CTRPv2 pan-cancer AAC 0.2 9e-08
mRNA MFSD11 CTRPv2 pan-cancer AAC 0.18 1e-07
mRNA AMPD1 CTRPv2 pan-cancer AAC 0.18 1e-07
mRNA FGFR3 CTRPv2 pan-cancer AAC 0.18 1e-07
mRNA LINGO1 CTRPv2 pan-cancer AAC 0.19 1e-07
mRNA RFTN1 CTRPv2 pan-cancer AAC -0.19 1e-07
mRNA FAM134C CTRPv2 pan-cancer AAC 0.18 1e-07
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