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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA PIGM CTRPv2 pan-cancer AAC 0.2 5e-09
mRNA TOR2A CTRPv2 pan-cancer AAC 0.21 5e-09
mRNA IREB2 GDSC1000 pan-cancer AAC 0.21 5e-09
mRNA FANCF CTRPv2 pan-cancer AAC 0.21 6e-09
mRNA STX7 CTRPv2 pan-cancer AAC -0.21 7e-09
mRNA LILRB4 CTRPv2 pan-cancer AAC 0.2 8e-09
mRNA DERL3 CTRPv2 pan-cancer AAC 0.2 8e-09
mRNA INSR CTRPv2 pan-cancer AAC 0.21 1e-08
mRNA KLF13 CTRPv2 pan-cancer AAC 0.22 1e-08
mRNA CD28 CTRPv2 pan-cancer AAC 0.2 1e-08
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