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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA HPCA CTRPv2 pan-cancer AAC 0.15 1e-05
mRNA ATXN7L3B CTRPv2 pan-cancer AAC 0.16 1e-05
mRNA TLE3 CTRPv2 pan-cancer AAC 0.15 1e-05
mRNA ARHGAP45 CTRPv2 pan-cancer AAC 0.22 1e-05
mRNA PAXIP1 CTRPv2 pan-cancer AAC 0.16 1e-05
mRNA C11orf68 CTRPv2 pan-cancer AAC -0.15 1e-05
mRNA GRIFIN CTRPv2 pan-cancer AAC 0.15 1e-05
mRNA MAML1 GDSC1000 pan-cancer AAC 0.14 1e-05
mRNA C1orf43 CTRPv2 pan-cancer AAC 0.16 1e-05
mRNA FRAT2 GDSC1000 pan-cancer AAC 0.16 1e-05
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