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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA UBN2 CTRPv2 pan-cancer AAC 0.17 6e-06
mRNA BCAS4 CTRPv2 pan-cancer AAC -0.16 6e-06
mRNA CERS6 CTRPv2 pan-cancer AAC 0.16 7e-06
mRNA TMEM97 CTRPv2 pan-cancer AAC 0.16 7e-06
mRNA CTDSP1 GDSC1000 pan-cancer AAC 0.16 7e-06
mRNA SRPRB CTRPv2 pan-cancer AAC 0.15 7e-06
mRNA TP53INP1 CTRPv2 pan-cancer AAC 0.16 7e-06
mRNA C1orf21 CTRPv2 pan-cancer AAC 0.16 7e-06
mRNA TRIM5 CTRPv2 pan-cancer AAC -0.16 7e-06
mRNA AMER2 CTRPv2 pan-cancer AAC 0.16 7e-06
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