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BMS-754807

Synonyms

SourcesNames Used
GDSC1000, FIMM, CTRPv2BMS-754807
PharmacoGx BMS-754807

External IDs

DatabaseIdentifier
Smiles: CC1(CCCN1C2=NN3C=CC=C3C(=N2)NC4=NNC(=C4)C5CC5)C(=O)NC6=CN=C(C=C6)F
Inchikey: LQVXSNNAFNGRAH-QHCPKHFHSA-N
Pubchem: 24785538

Annotated Targets

INSR, IGF1R, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BMS-754807


Feature TypeStandardized
Nominal ANOVA
mRNA GRHPR CTRPv2 pan-cancer AAC -0.16 3e-06
mRNA POLE3 CTRPv2 pan-cancer AAC 0.17 3e-06
mRNA KDM7A CTRPv2 pan-cancer AAC 0.17 3e-06
mRNA CBX2 CTRPv2 pan-cancer AAC 0.18 3e-06
mRNA ACAP3 CTRPv2 pan-cancer AAC 0.16 3e-06
mRNA KCNA3 CTRPv2 pan-cancer AAC 0.18 3e-06
mRNA SIGMAR1 CTRPv2 pan-cancer AAC 0.16 3e-06
mRNA MSTO1 CTRPv2 pan-cancer AAC 0.16 3e-06
mRNA GPX8 CTRPv2 pan-cancer AAC -0.2 4e-06
mRNA GLB1L2 CTRPv2 pan-cancer AAC 0.18 4e-06
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