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PD-0325901

Synonyms

SourcesNames Used
CCLE, GDSC1000PD-0325901
gCSIpd0325901
PharmacoGx PD-0325901

External IDs

DatabaseIdentifier
Smiles: C1=CC(=C(C=C1I)F)NC2=C(C=CC(=C2F)F)C(=O)NOCC(CO)O
Inchikey: SUDAHWBOROXANE-SECBINFHSA-N
Pubchem: 9826528

Annotated Targets

MAP2K1, MAP2K2

FDA Approval Status

Not Approved
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Top molecular features associated with response to PD-0325901


Feature TypeStandardized
Nominal ANOVA
mRNA MAP4K1 gCSI pan-cancer AAC -0.51 6e-09
mRNA IKZF1 CCLE pan-cancer AAC -0.49 8e-08
mRNA TCF4 gCSI pan-cancer AAC -0.43 1e-11
mRNA POU2AF1 gCSI pan-cancer AAC -0.43 4e-09
mRNA ATP6V1G2 gCSI pan-cancer AAC -0.42 3e-12
mRNA CARMIL2 gCSI pan-cancer AAC -0.4 8e-11
mRNA LRMP gCSI pan-cancer AAC -0.4 2e-06
mRNA SEPT1 gCSI pan-cancer AAC -0.4 6e-10
mRNA MAP4K1 CCLE pan-cancer AAC -0.39 2e-08
mRNA RUNX1T1 gCSI pan-cancer AAC -0.39 3e-13
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