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tissues
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cell lines
23132-87
AGS
AZ-521
BGC-823
ECC10
ECC12
FU97
GCIY
GSS
GSU
GT3TKB
GTL-16
HGC-27
Hs 746T
HSC-39
HuG1-N
IM-95
IM-95m
KATOIII
KE-39
LMSU
MKN1
MKN28
MKN45
MKN7
MKN74
NCC-StC-K140
NCI-N87
NCI-SNU-1
NCI-SNU-16
NCI-SNU-5
NUGC-2
NUGC-3
NUGC-4
OCUM-1
Okajima
RERF-GC-1B
RF-48
SCH
SH-10-TC
SNU-1
SNU-16
SNU-216
SNU-484
SNU-5
SNU-520
SNU-601
SNU-620
SNU-638
SNU-668
SNU-719
Takigawa
TGBC11TKB
TMK-1
drugs
AEW541
Nilotinib
17-AAG
PHA-665752
lapatinib
Nutlin-3
AZD0530
Crizotinib
L-685458
Vandetanib
Panobinostat
Sorafenib
Irinotecan
Topotecan
LBW242
PD-0325901
PD-0332991
paclitaxel
AZD6244
PLX4720
RAF265
TAE684
TKI258
Erlotinib
JQ12
XMD15-27
VNLG/124
LFM-A13
AZD6482
GSK2126458
TG-101348
FH535
STF-62247
SB52334
KIN001-260
FR-180204
AS601245
XMD13-2
Genentech Cpd 10
Obatoclax Mesylate
XMD14-99
VX-11e
EKB-569
ZSTK474
AS605240
KIN001-270
T0901317
NSC-87877
Bryostatin 1
KIN001-244
Bleomycin
LAQ824
AKT inhibitor VIII
PF-562271
CH5424802
NSC-207895
GSK-650394
AC220
foretinib
BX-912
Mitomycin-C
LY317615
tivozanib
Zibotentan
CP466722
HG-6-64-1
CHIR-99021
BMS-754807
GSK-1904529A
GSK1070916
KIN001-266
masitinib
Ispinesib Mesylate
pac-1
JQ-1
ruxolitinib
FTI-277
QL-X-138
OSI-930
CX-5461
SNX-2112
OSI-027
Vinorelbine
JW-7-24-1
Epothilone B
BMS-345541
FMK
BIX02189
Bicalutamide
Salubrinal
Lisitinib
etoposide
WZ3105
MS-275
WH-4-023
Doxorubicin
linifanib
BMS-509744
embelin
KIN001-102
Bexarotene
DMOG
JNK-9L
PI-103
KIN001-135
GSK429286A
GSK690693
Bortezomib
Pazopanib
Parthenolide
NPK76-II-72-1
MP470
OSU-03012
shikonin
Cyclopamine
MPS-1-IN-1
QS11
AR-42
TGX221
PHA-793887
QL-XII-47
KIN001-236
NG-25
Z-LLNle-CHO
CMK
TAK-715
GW843682X
BHG712
KIN001-055
GW-2580
BAY 61-3606
Gemcitabine
BMS-536924
TL-2-105
AZ628
AUY922
GSK269962A
AT-7519
CP724714
A-443654
JW-7-52-1
IPA-3
phenformin
Imatinib
MG-132
UNC0638
PIK-93
belinostat
5-FU
THZ-2-49
Roscovitine
TL-1-85
QL-XI-92
BMS-708163
Y-39983
GNF-2
S-Trityl-L-cysteine
Sunitinib
CUDC-101
Midostaurin
Pyrimethamine
CAY10603
BI-2536
Rapamycin
CGP-082996
CAL-101
YM-155
Tipifarnib
XL-184
CGP-60474
I-BET-762
tubastatin A
thapsigargin
THZ-2-102-1
WZ-1-84
XMD8-85
AP-24534
YM201636
Dasatinib
EX-527
VX-680
TPCA-1
A-770041
BIBW2992
dabrafenib
IOX2
Cisplatin
ATRA
KU-55933
AG-014699
MK-2206
AICAR
JNJ-26854165
TW 37
Cytarabine
681640
FK866
Tamoxifen
GW 441756
(5Z)-7-Oxozeaenol
Bosutinib
ABT-263
XAV-939
PF-4708671
Cetuximab
piperlongumine
PFI-1
AZD7762
MLN4924
Methotrexate
NVP-BEZ235
SB590885
AZD-2281
CI-1040
SB 216763
Talazoparib
AZD8055
Vinblastine
PD173074
lenalidomide
NU-7441
VX-702
SN-38
UNC1215
Camptothecin
GDC-0941
BIRB 0796
CCT018159
JNK Inhibitor VIII
RO-3306
ABT-888
RDEA119
BX-795
SGC0946
GSK1120212
rTRAIL
GDC-0449
temozolomide
Elesclomol
ZM-447439
temsirolimus
SB 505124
Nutlin-3a (-)
CEP-701
XMD8-92
HG-5-113-01
XMD11-85h
CCT007093
Gefitinib
ZG-10
AMG-706
SL 0101-1
Docetaxel
Vorinostat
Axitinib
QL-VIII-58
EHT 1864
HG-5-88-01
QL-XII-61
YK 4-279
bid1870
CIL55
BRD4132
BRD6340
ML006
Bax channel blocker
BRD9876
betulinic acid
phloretin
gossypol
chlorambucil
isoliquiritigenin
cimetidine
azacitidine
trifluoperazine
Carboplatin
Teniposide
Sildenafil
simvastatin
parbendazole
procarbazine
Curcumin
ciclopirox
myricetin
lovastatin
valdecoxib
dacarbazine
prochlorperazine
ifosfamide
ouabain
BRD9647
BRD-K26531177
NSC23766
pyrazolanthrone
C6-ceramide
N9-isopropylolomoucine
importazole
prima-1
blebbistatin
cytochalasin b
NSC95397
manumycin A
tacrolimus
pifithrin-alpha
SB-431542
staurosporine
SB-225002
Cerulenin
purmorphamine
GSK-3 inhibitor IX
BRD-K94991378
BIX-01294
IC-87114
ciclosporin
sitagliptin
PDMP
BRD-K71935468
BEC
apicidin
Merck60
BRD-A94377914
FGIN-1-27
compound 1B
vincristine
itraconazole
erastin
ML031
CIL56
FQI-1
BRD-K92856060
B02
BRD-K45681478
ML050
ML162
CIL41
NSC30930
CIL70
MI-1
DBeQ
ML083
CID-5951923
IU1
dexamethasone
ML311
decitabine
BRD-K61166597
CHEMBL374350
QW-BI-011
bendamustine
CD-437
SCH-79797
LE-135
SKI-II
CI-976
Platin
necrostatin-1
GW-405833
AC55649
RITA
LY-2183240
CD-1530
NSC632839
pifithrin-mu
BRD-K80183349
BRD-K66532283
triazolothiadiazine
BRD-K66453893
BRD-K11533227
BRD-K27224038
BRD-K14844214
BRD1835
BRD-K41597374
BRD-K63431240
BRD-K13999467
BRD-K96970199
brefeldin A
AGK-2
PF-750
triptolide
AA-COCF3
16-beta-bromoandrosterone
PRL-3 Inhibitor I
SID 26681509
CHEMBL1222381
NSC 74859
ABT-737
Zebularine
SR-II-138A
Compound 7d-cis
AZD-7545
VER-155008
ML203
SRT-1720
CAY10594
Compound 1541A
RG-108
pluripotin
GMX-1778
MST-312
oligomycin a
indisulam
BRD-K49290616
BRD-K02492147
austocystin d
SJ-172550
BRD-K09587429
pandacostat
BRD-K96431673
cyanoquinoline 11
tipifarnib
Compound 23 citrate
nakiterpiosin
CCT036477
tamatinib
myriocin
BIBR-1532
neratinib
BRD1812
BRD8958
MK 1775
Ko-143
CR-1-31B
BRD-K71781559
BRD-K86535717
BRD-K48334597
ML312
BRD-K04800985
BRD-K78574327
BRD-K19103580
BRD-K30019337
BRD-K84807411
BRD-K44224150
BRD-K75293299
BRD-K64610608
BRD-K02251932
BRD-K55116708
BRD-K41334119
BRD-K34485477
BRD-K16147474
BRD-K29086754
BRD-K33199242
BRD-K52037352
BRD-K27986637
BRD-K37390332
tandutinib
fulvestrant
HLI 373
NSC48300
PRIMA-1-Met
isoevodiamine
cucurbitacin I
BRD-K50799972
BRD-K17060750
canertinib
brivanib
GDC-0879
SNS-032
KU-0063794
TG-100-115
SU11274
BRD-K88742110
BRD8899
ELCPK
NPC-26
1S,3R-RSL-3
CIL55A
SCH-529074
StemRegenin 1
FQI-2
ML210
darinaparsin
PX-12
GANT-61
PL-DI
CHM-1
ML239
Fumonisin B1
BRD-K51490254
BRD-K85133207
CAY10576
Repligen 136
nintedanib
regorafenib
WZ8040
MGCD-265
lenvatinib
CAY10618
KU 0060648
narciclasine
MLN2238
ISOX
BRD-K29313308
UNC0321
SGX-523
erismodegib
alisertib
SB-525334
quizartinib
fingolimod
pazopanib
BRD-K24690302
BRD-K70511574
PLX-4032
GSK461364
BRD-K20514654
BRD-K28456706
STF-31
spautin-1
BRD-A02303741
ML320
tigecycline
PF-543
PF-573228
ceranib-2
FSC231
968
GSK4112
etomoxir
HC-067047
IPR-456
leptomycin B
AZ-3146
VU0155056
JQ-1:UNC0638 (2:1 mol/mol)
carboplatin:UNC0638 (2:1 mol/mol)
vorinostat:carboplatin (1:1 mol/mol)
serdemetan:SCH-529074 (1:1 mol/mol)
selumetinib:PLX-4032 (8:1 mol/mol)
sirolimus:bortezomib (250:1 mol/mol)
BRD-K97651142
vorapaxar
Ch-55
BRD-K79669418
BRD-K99584050
BRD-A71883111
navitoclax:birinapant (1:1 mol/mol)
ISOX:bortezomib (250:1 mol/mol)
selumetinib:GDC-0941 (4:1 mol/mol)
selumetinib:tretinoin (2:1 mol/mol)
selumetinib:vorinostat (8:1 mol/mol)
selumetinib:JQ-1 (4:1 mol/mol)
selumetinib:BRD-A02303741 (4:1 mol/mol)
tretinoin:navitoclax (4:1 mol/mol)
decitabine:navitoclax (2:1 mol/mol)
tretinoin:carboplatin (2:1 mol/mol)
necrostatin-7
PYR-41
I-BET151
lomeguatrib
tanespimycin:gemcitabine (1:1 mol/mol)
docetaxel:tanespimycin (2:1 mol/mol)
selumetinib:MK-2206 (8:1 mol/mol)
navitoclax:PLX-4032 (1:1 mol/mol)
selumetinib:piperlongumine (8:1 mol/mol)
tanespimycin:bortezomib (250:1 mol/mol)
navitoclax:MST-312 (1:1 mol/mol)
carboplatin:etoposide (40:17 mol/mol)
piperlongumine:MST-312 (1:1 mol/mol)
navitoclax:gemcitabine (1:1 mol/mol)
JW-480
BMS-195614
BRD-K07442505
BRD-K35604418
SB-743921
GSK525762A
navitoclax:pluripotin (1:1 mol/mol)
JQ-1:carboplatin (1:1 mol/mol)
selumetinib:navitoclax (8:1 mol/mol)
selumetinib:decitabine (4:1 mol/mol)
decitabine:carboplatin (1:1 mol/mol)
SNX-2112:bortezomib (250:1 mol/mol)
JQ-1:navitoclax (2:1 mol/mol)
JQ-1:MK-0752 (1:1 mol/mol)
BRD-A02303741:navitoclax (2:1 mol/mol)
salermide:PLX-4032 (12:1 mol/mol)
UNC0638:navitoclax (1:1 mol/mol)
BRD-A02303741:carboplatin (1:1 mol/mol)
doxorubicin:navitoclax (2:1 mol/mol)
selumetinib:UNC0638 (4:1 mol/mol)
alisertib:navitoclax (2:1 mol/mol)
navitoclax:sorafenib (1:1 mol/mol)
navitoclax:piperlongumine (1:1 mol/mol)
SMER-3
NVP-ADW742
clofarabine
vorinostat:navitoclax (4:1 mol/mol)
XL765
ML258
SR1001
bardoxolone methyl
elocalcitol
BMS-270394
fluvastatin
AZD4547
hyperforin
NVP-231
MK-0752
semagacestat
nelarabine
rigosertib
PD318088
KU-60019
KW-2449
silmitasertib
BRD-K03911514
BRD-K16130065
momelotinib
LY-2157299
WP1130
NVP-BSK805
erlotinib:PLX-4032 (2:1 mol/mol)
birinapant
KX2-391
3-Cl-AHPC
BRD-K58730230
BRD-K27188169
KHS101
WAY-362450
JQ-1:vorinostat (2:1 mol/mol)
BRD-K13185470
cabozantinib
crizotinib:PLX-4032 (2:1 mol/mol)
BRD-K27188169:navitoclax (2:1 mol/mol)
BRD-K03536150
BRD-K34222889
OSI-906
epigallocatechin-3-monogallate
Cyclophosphamide
niclosamide
AM-580
Mdivi-1
Ki8751
Oxaliplatin
neopeltolide
tosedostat
barasertib
YL54
BRD-K34099515
PF-184
AT7867
PD 153035
tacedinaline
omacetaxine mepesuccinate
avrainvillamide
BRD-K09344309
isonicotinohydroxamic acid
NSC19630
LRRK2-IN-1
salermide
WZ4002
ML334 diastereomer
KH-CB19
abiraterone
KPT185
pitstop2
R428
ibrutinib
sotrastaurin
A-804598
COL-3
ABT-199
ETP-46464
marinopyrrole A
methylstat
BYL-719
GSK2636771
necrosulfonamide
HBX-41108
palmostatin B
JW-55
AT-406
JW-74
GSK1059615
BRD-K55473186
VAF-347
BRD-M00053801
thalidomide
O-6-benzylguanine
BRD-K90370028
cediranib
BRD-K48477130
AZD1480
BRD-A05715709
BRD-K99006945
tivantinib
RO4929097
dinaciclib
MLN2480
BRD-K51831558
istradefylline
MI-2
BRD-K42260513
alvocidib
CBB-1007
BRD-A86708339
PF-3758309
SZ4TA2
AT13387
BCL-LZH-4
skepinone-L
PF-4800567 hydrochloride
avicin D
BRD-K33514849
BRD-K01737880
bafilomycin A1
SR8278
GSK-J4
BRD9876:MK-1775 (4:1 mol/mol)
BRD-K30748066
targets
ABAT
ABCB1
ABCC1
ABCG2
ABL1
ABL2
ACADSB
ACAT1
ACER1
ACER2
ACER3
ACHE
ACTB
ACVR1C
ADORA1
ADORA2A
ADORA2B
ADORA3
ADRA1A
AHR
AKT1
AKT2
AKT3
ALDH2
ALDH5A1
ALK
ALOX5
ANPEP
ANXA1
APH1A
APP
AQP9
AR
ARAF
ARF1
ARFGAP1
ARG1
ARG2
ASAH1
ASAH2
ASAH2B
ATIC
ATM
ATP1A1
ATP1A2
ATP1A3
ATP1A4
ATP1B1
ATP1B2
ATP1B3
ATP1B4
ATP5A1
ATP5L2
ATP6V0A1
ATP6V1A
ATR
AURKA
AURKB
AURKC
AXL
BAD
BAX
BCL2
BCL2L1
BCL2L10
BCL2L2
BCR
BIRC2
BIRC5
BLK
BMX
BRAF
BRD2
BRD3
BRD4
BRDT
BTK
C1QA
C1QB
C1QC
C1R
C1S
CA1
CA12
CA14
CA2
CA4
CA6
CA7
CA9
CALM1
CALY
CAMK1D
CAMK2G
CASP3
CASP6
CASP7
CCNA2
CCNB1
CCNE1
CDA
CDC25A
CDC25B
CDC25C
CDH5
CDK1
CDK14
CDK16
CDK17
CDK2
CDK4
CDK5
CDK5R1
CDK6
CDK7
CDK8
CDK9
CDKL5
CENPE
CERK
CERS1
CERS2
CERS3
CERS4
CERS5
CERS6
CES1
CHD1
CHEK1
CHEK2
CHUK
CLCN3
CLK1
CLK3
CLK4
CLTA
CLTB
CLTC
CLTCL1
CMPK1
CNR2
CPT1A
CRBN
CSF1
CSF1R
CSK
CSNK1D
CSNK1E
CSNK1G3
CSNK2A1
CSNK2A2
CUL1
CXCR2
CYP11B1
CYP17A1
CYP2A6
CYP2B6
CYP2C18
CYP2C19
CYP2C8
CYP2C9
CYP2D6
CYP3A4
CYP3A5
CYP3A7
CYP51A1
CYTH2
DBH
DCLK1
DCLK2
DDR1
DDR2
DHFR
DHX9
DIABLO
DNM1
DNMT1
DNMT3A
DNMT3B
DOT1L
DPP4
DRD1
DRD2
DRD3
DRD4
DYRK1A
EBP
EDNRA
EGFR
EGLN1
EHMT1
EHMT2
EIF2S1
EIF4A2
EIF4E
EIF4G1
EP300
EPHA1
EPHA10
EPHA2
EPHA3
EPHA4
EPHA5
EPHA6
EPHA7
EPHA8
EPHB1
EPHB2
EPHB3
EPHB4
EPHB6
ERBB2
ERBB3
ERBB4
ERG
ESR1
ESR2
ETV1
EWSR1
EZH2
F2R
FAAH
FASN
FCGR1A
FCGR2A
FCGR2B
FCGR3A
FCGR3B
FGF1
FGFR1
FGFR2
FGFR3
FGFR4
FGR
FKBP1A
FLI1
FLT1
FLT3
FLT4
FNTA
FNTB
FRK
FYN
GABBR1
GART
GLO1
GLS
GPBAR1
GPER1
GSK3A
GSK3B
HCK
HDAC1
HDAC10
HDAC11
HDAC2
HDAC3
HDAC4
HDAC5
HDAC6
HDAC7
HDAC8
HDAC9
HMGCR
HMGCS1
HNF4A
HRH1
HRH2
HSP90AA1
HSP90AB1
HSP90B1
HSPA1A
HSPA1B
HSPA1L
HTR2A
HTR2C
IDH1
IGF1R
IKBKB
IKBKE
IL1B
IL6
INSR
ITGAL
ITGB2
ITK
JAK1
JAK2
JAK3
JUN
KCNH2
KCNJ8
KDM1A
KDM2A
KDM3A
KDM4A
KDM4B
KDM4C
KDM4D
KDM5C
KDM6A
KDM6B
KDR
KEAP1
KIF11
KIT
KLF5
KPNB1
L3MBTL3
LAP3
LCK
LDHA
LDHB
LDHC
LIG1
LIG3
LIMK1
LRRK2
LYN
LYPLA1
MAP2
MAP2K1
MAP2K2
MAP2K5
MAP3K2
MAP3K8
MAP4
MAP4K5
MAPK1
MAPK11
MAPK12
MAPK14
MAPK3
MAPK7
MAPK8
MAPKAPK2
MAPT
MCL1
MDM2
MDM4
MEN1
MET
MGMT
MMP13
MMP9
MST1R
MTOR
MYH1
MYH2
NAMPT
NCEH1
NCOA1
NCOA2
NCSTN
NEK11
NFE2L2
NFKB1
NOS2
NPEPPS
NPM1
NR0B1
NR0B2
NR1D1
NR1H2
NR1H3
NR1H4
NR1I2
NR3C1
NR3C2
NTRK1
OGDH
ORM1
ORM2
P2RX7
PAK1
PAK4
PAK6
PARP1
PARP2
PARP3
PDE4A
PDE4B
PDE4D
PDE5A
PDE6G
PDE6H
PDGFD
PDGFRA
PDGFRB
PDK1
PDK2
PDPK1
PGD
PI4KB
PICK1
PIK3C3
PIK3CA
PIK3CB
PIK3CD
PIK3CG
PIM1
PKIA
PKM
PLA2G4A
PLA2G4B
PLA2G4C
PLA2G4D
PLAUR
PLD1
PLD2
PLK1
PLK2
PLK3
PLK4
POLA1
POLA2
POLB
POLD1
POLE
PPID
PPP2CA
PPP3CA
PPP3CB
PPP3CC
PPP3R1
PPP3R2
PREP
PRKAA1
PRKACA
PRKACB
PRKCA
PRKCB
PRKCD
PRKCE
PRKCG
PRKCH
PRKCI
PRKCQ
PRKCZ
PRKDC
PRKG1
PRKX
PSEN1
PSENEN
PSMA1
PSMA2
PSMA3
PSMA4
PSMA5
PSMA6
PSMA7
PSMA8
PSMB1
PSMB10
PSMB11
PSMB2
PSMB3
PSMB4
PSMB5
PSMB6
PSMB7
PSMB8
PSMB9
PSMD1
PSMD2
PTGS1
PTGS2
PTK2
PTK2B
PTK6
PTP4A3
PYGM
RAC1
RAD51
RAF1
RARA
RARB
RARG
RASAL1
RELA
RET
RHOA
RIPK1
ROCK1
ROCK2
RORA
RORC
RPS6KA1
RPS6KA2
RPS6KA3
RPS6KA6
RPS6KB1
RPS6KB2
RRM1
RRM2
RRM2B
RXRA
RXRB
RXRG
S100A4
S1PR1
S1PR3
S1PR5
SCARB1
SCN10A
SCN11A
SCN1A
SCN1B
SCN2A
SCN2B
SCN3A
SCN3B
SCN4A
SCN4B
SCN5A
SCN7A
SCN8A
SCN9A
SELL
SELP
SENP2
SGK1
SGK2
SH2B3
SIK1
SIRT1
SIRT2
SKP1
SLC23A1
SLC29A4
SLC47A1
SLC47A2
SLC5A1
SLC7A11
SLCO1B1
SLCO1B3
SMO
SPHK1
SPTLC1
SPTLC2
SPTLC3
SRC
SRD5A2
SRMS
STAT3
STAT5B
STK10
STK24
STK33
STK4
SYK
TACC3
TASP1
TEK
TERT
TGFBR1
TIAM1
TLR4
TNF
TNFSF11
TNK1
TNK2
TNKS
TNKS2
TNNC1
TOP1
TOP1MT
TOP2A
TOP2B
TP53
TRIO
TRPC6
TRPV4
TSPO
TTK
TUBA1A
TUBA1B
TUBA1C
TUBA3C
TUBA3D
TUBA3E
TUBA4A
TUBA8
TUBB
TUBB1
TUBB2A
TUBB2B
TUBB3
TUBB4A
TUBB4B
TUBB6
TUBB8
TUBD1
TUBE1
TUBG1
TXK
TXN
TXNRD1
TYK2
TYMS
UCHL5
UGCG
USP1
USP10
USP13
USP14
USP2
USP5
USP7
USP9X
VCP
VDAC1
VDAC2
VDR
VEGFA
WEE1
XDH
XIAP
XPO1
YES1
ZAP70