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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA EVL CTRPv2 pan-cancer AAC 0.23 8e-12
mRNA ATAD5 CTRPv2 pan-cancer AAC 0.24 9e-12
mRNA ZBTB3 CTRPv2 pan-cancer AAC 0.24 9e-12
mRNA PDS5B CTRPv2 pan-cancer AAC 0.23 1e-11
mRNA TMPO CTRPv2 pan-cancer AAC 0.23 1e-11
mRNA LAT2 CTRPv2 pan-cancer AAC 0.25 1e-11
mRNA PIKFYVE CTRPv2 pan-cancer AAC 0.26 1e-11
mRNA NUDT3 CTRPv2 pan-cancer AAC 0.25 1e-11
mRNA ZBED3 CTRPv2 pan-cancer AAC 0.23 2e-11
mRNA KANSL1 CTRPv2 pan-cancer AAC 0.23 2e-11
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