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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA LINGO2 CTRPv2 pan-cancer AAC 0.12 0.0004
mRNA TNFAIP8L2 CTRPv2 pan-cancer AAC 0.14 0.0004
mRNA CD3E CTRPv2 pan-cancer AAC 0.11 0.0004
mRNA SPSB1 CTRPv2 pan-cancer AAC -0.12 0.0004
mRNA GOSR2 CTRPv2 pan-cancer AAC -0.12 0.0004
mRNA SNRK CTRPv2 pan-cancer AAC 0.12 0.0004
mRNA AF011889.5 CTRPv2 pan-cancer AAC -0.12 0.0004
mRNA C16orf54 CTRPv2 pan-cancer AAC 0.13 0.0004
mRNA C19orf68 CTRPv2 pan-cancer AAC 0.11 0.0004
mRNA NKX6-1 CTRPv2 pan-cancer AAC 0.12 0.0004
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