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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA GMFG CTRPv2 pan-cancer AAC 0.39 3e-17
mRNA MBTD1 CTRPv2 pan-cancer AAC 0.36 4e-21
mRNA WAS CTRPv2 pan-cancer AAC 0.35 4e-09
mRNA CBX2 CTRPv2 pan-cancer AAC 0.35 5e-23
mRNA NCKAP1L CTRPv2 pan-cancer AAC 0.34 2e-13
mRNA CDCA7 CTRPv2 pan-cancer AAC 0.34 2e-22
mRNA ZBED4 CTRPv2 pan-cancer AAC 0.34 5e-20
mRNA ARHGAP19 CTRPv2 pan-cancer AAC 0.33 9e-17
mRNA GRK2 CTRPv2 pan-cancer AAC 0.33 9e-16
mRNA CTB-133G6.1 CTRPv2 pan-cancer AAC 0.33 2e-17
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