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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA MED28 CTRPv2 pan-cancer AAC 0.3 4e-14
mRNA RASGRP2 CTRPv2 pan-cancer AAC 0.3 3e-14
mRNA FBRSL1 CTRPv2 pan-cancer AAC 0.29 1e-18
mRNA ZNF445 CTRPv2 pan-cancer AAC 0.29 7e-16
mRNA TFAP4 CTRPv2 pan-cancer AAC 0.29 4e-16
mRNA CNOT8 CTRPv2 pan-cancer AAC 0.29 5e-17
mRNA YPEL1 CTRPv2 pan-cancer AAC 0.29 9e-18
mRNA LMNB1 CTRPv2 pan-cancer AAC 0.29 2e-16
mRNA SCAF4 CTRPv2 pan-cancer AAC 0.29 6e-15
mRNA CNTRL CTRPv2 pan-cancer AAC 0.29 2e-11
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