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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA GMIP CTRPv2 pan-cancer AAC 0.25 3e-09
mRNA H3F3A CTRPv2 pan-cancer AAC 0.21 3e-09
mRNA MAZ CTRPv2 pan-cancer AAC 0.2 3e-09
mRNA PIDD1 CTRPv2 pan-cancer AAC 0.2 3e-09
mRNA IRF2BP2 CTRPv2 pan-cancer AAC 0.2 3e-09
mRNA PBRM1 CTRPv2 pan-cancer AAC 0.21 3e-09
mRNA GPC2 CTRPv2 pan-cancer AAC 0.24 3e-09
mRNA C7orf55-LUC7L2 CTRPv2 pan-cancer AAC 0.21 3e-09
mRNA DNMT1 CTRPv2 pan-cancer AAC 0.22 3e-09
mRNA SRRT CTRPv2 pan-cancer AAC 0.2 3e-09
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