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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA GRAMD1A CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA MBNL3 CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA SYT1 CTRPv2 pan-cancer AAC 0.14 0.0002
mRNA H1FX CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA FDFT1 CTRPv2 pan-cancer AAC 0.13 0.0002
mRNA WWOX CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA ATP6V1D CTRPv2 pan-cancer AAC -0.13 0.0002
mRNA KRT72 CTRPv2 pan-cancer AAC 0.11 0.0002
mRNA BTD CTRPv2 pan-cancer AAC -0.13 0.0002
mRNA ZNF571 CTRPv2 pan-cancer AAC 0.12 0.0002
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