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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA CTD-2207O23.3 CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA PRDM16 CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA TDG CTRPv2 pan-cancer AAC 0.13 0.0002
mRNA KANSL3 CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA SDHB CTRPv2 pan-cancer AAC -0.12 0.0002
mRNA ZNF605 CTRPv2 pan-cancer AAC 0.13 0.0002
mRNA U2AF2 CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA MBD3L3 CTRPv2 pan-cancer AAC 0.13 0.0002
mRNA RP11-96L14.7 CTRPv2 pan-cancer AAC -0.12 0.0002
mRNA PIK3C3 CTRPv2 pan-cancer AAC 0.13 0.0002
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