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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA ZNF783 CTRPv2 pan-cancer AAC 0.13 0.0002
mRNA RBL2 CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA ZNF280C CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA C15orf61 CTRPv2 pan-cancer AAC 0.13 0.0002
mRNA SLC43A1 CTRPv2 pan-cancer AAC 0.14 0.0002
mRNA TMEM115 CTRPv2 pan-cancer AAC -0.14 0.0002
mRNA CEBPG CTRPv2 pan-cancer AAC 0.13 0.0002
mRNA LAMC1 CTRPv2 pan-cancer AAC -0.14 0.0002
mRNA ZFP90 CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA USP13 CTRPv2 pan-cancer AAC 0.12 0.0002
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