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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA TRIM65 CTRPv2 pan-cancer AAC 0.22 2e-10
mRNA LPAR2 CTRPv2 pan-cancer AAC 0.22 2e-10
mRNA BEND3 CTRPv2 pan-cancer AAC 0.22 2e-10
mRNA EP400 CTRPv2 pan-cancer AAC 0.21 2e-10
mRNA RP11-15H20.8 CTRPv2 pan-cancer AAC 0.21 2e-10
mRNA CBX8 CTRPv2 pan-cancer AAC 0.22 2e-10
mRNA TTF1 CTRPv2 pan-cancer AAC 0.21 2e-10
mRNA C20orf96 CTRPv2 pan-cancer AAC 0.21 2e-10
mRNA S1PR4 CTRPv2 pan-cancer AAC 0.24 2e-10
mRNA TAF5 CTRPv2 pan-cancer AAC 0.23 2e-10
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