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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA RNASEH2B CTRPv2 pan-cancer AAC 0.25 7e-11
mRNA CXCR4 CTRPv2 pan-cancer AAC 0.24 7e-11
mRNA HNRNPDL CTRPv2 pan-cancer AAC 0.23 8e-11
mRNA CDT1 CTRPv2 pan-cancer AAC 0.25 8e-11
mRNA NFATC3 CTRPv2 pan-cancer AAC 0.27 8e-11
mRNA PARVG CTRPv2 pan-cancer AAC 0.23 8e-11
mRNA CTCF CTRPv2 pan-cancer AAC 0.24 8e-11
mRNA PNISR CTRPv2 pan-cancer AAC 0.22 9e-11
mRNA FCHO1 CTRPv2 pan-cancer AAC 0.28 1e-10
mRNA TEX22 CTRPv2 pan-cancer AAC 0.22 1e-10
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