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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA ADGRL1 CTRPv2 pan-cancer AAC 0.23 3e-11
mRNA KHDRBS1 CTRPv2 pan-cancer AAC 0.22 3e-11
mRNA ABHD17B CTRPv2 pan-cancer AAC 0.22 3e-11
mRNA SLC35E2 CTRPv2 pan-cancer AAC 0.22 4e-11
mRNA RSBN1 CTRPv2 pan-cancer AAC 0.23 4e-11
mRNA LRRC37A2 CTRPv2 pan-cancer AAC 0.22 5e-11
mRNA CASP8AP2 CTRPv2 pan-cancer AAC 0.22 5e-11
mRNA PDE7A CTRPv2 pan-cancer AAC 0.24 6e-11
mRNA ARHGAP45 CTRPv2 pan-cancer AAC 0.3 6e-11
mRNA SUGP1 CTRPv2 pan-cancer AAC 0.22 6e-11
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