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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA CTD-2207O23.12 CTRPv2 pan-cancer AAC 0.13 0.0003
mRNA BUB1B CTRPv2 pan-cancer AAC 0.12 0.0003
mRNA ST20-MTHFS CTRPv2 pan-cancer AAC -0.11 0.0003
mRNA GPRIN1 CTRPv2 pan-cancer AAC 0.12 0.0003
mRNA RP11-12J10.3 CTRPv2 pan-cancer AAC 0.12 0.0003
mRNA CHKB CTRPv2 pan-cancer AAC 0.12 0.0003
mRNA HSD3B7 CTRPv2 pan-cancer AAC -0.12 0.0003
mRNA GPR173 CTRPv2 pan-cancer AAC 0.15 0.0003
mRNA XAB2 CTRPv2 pan-cancer AAC 0.13 0.0003
mRNA ZNF704 CTRPv2 pan-cancer AAC 0.13 0.0003
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