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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA TBC1D24 CTRPv2 pan-cancer AAC 0.12 0.0003
mRNA GLUL CTRPv2 pan-cancer AAC 0.12 0.0003
mRNA AGO3 CTRPv2 pan-cancer AAC 0.12 0.0003
mRNA ITGA4 CTRPv2 pan-cancer AAC 0.15 0.0003
mRNA TAF8 CTRPv2 pan-cancer AAC 0.12 0.0003
mRNA BFAR CTRPv2 pan-cancer AAC -0.13 0.0003
mRNA MRPL24 CTRPv2 pan-cancer AAC -0.12 0.0003
mRNA CNN3 CTRPv2 pan-cancer AAC -0.15 0.0003
mRNA LTB4R2 CTRPv2 pan-cancer AAC 0.12 0.0003
mRNA POLI CTRPv2 pan-cancer AAC 0.12 0.0003
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