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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA EXOSC6 CTRPv2 pan-cancer AAC 0.17 3e-07
mRNA TRABD CTRPv2 pan-cancer AAC 0.2 3e-07
mRNA VAV1 CTRPv2 pan-cancer AAC 0.26 3e-07
mRNA CBX5 CTRPv2 pan-cancer AAC 0.18 3e-07
mRNA NT5M CTRPv2 pan-cancer AAC 0.17 3e-07
mRNA NKD2 CTRPv2 pan-cancer AAC 0.17 3e-07
mRNA ADNP2 CTRPv2 pan-cancer AAC 0.17 3e-07
mRNA SETMAR CTRPv2 pan-cancer AAC 0.18 3e-07
mRNA KHSRP CTRPv2 pan-cancer AAC 0.18 3e-07
mRNA GMPPA CTRPv2 pan-cancer AAC -0.16 3e-07
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