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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA TP53 CTRPv2 pan-cancer AAC 0.17 2e-07
mRNA USP37 CTRPv2 pan-cancer AAC 0.17 2e-07
mRNA P2RY11 CTRPv2 pan-cancer AAC 0.18 2e-07
mRNA KIAA1143 CTRPv2 pan-cancer AAC 0.18 2e-07
mRNA RAD54L2 CTRPv2 pan-cancer AAC 0.19 2e-07
mRNA PXDC1 CTRPv2 pan-cancer AAC -0.19 2e-07
mRNA TET1 CTRPv2 pan-cancer AAC 0.18 2e-07
mRNA SATB1 CTRPv2 pan-cancer AAC 0.18 2e-07
mRNA ZC4H2 CTRPv2 pan-cancer AAC 0.17 2e-07
mRNA ADAMTS10 CTRPv2 pan-cancer AAC 0.17 2e-07
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