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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA MDN1 CTRPv2 pan-cancer AAC 0.2 2e-08
mRNA EIF6 CTRPv2 pan-cancer AAC -0.19 2e-08
mRNA TCERG1 CTRPv2 pan-cancer AAC 0.19 2e-08
mRNA IL17RA CTRPv2 pan-cancer AAC 0.18 2e-08
mRNA ITGAL CTRPv2 pan-cancer AAC 0.2 2e-08
mRNA ZNF266 CTRPv2 pan-cancer AAC 0.2 2e-08
mRNA N4BP2L1 CTRPv2 pan-cancer AAC 0.22 2e-08
mRNA SF3B1 CTRPv2 pan-cancer AAC 0.18 2e-08
mRNA PLEKHO1 CTRPv2 pan-cancer AAC 0.2 2e-08
mRNA RP4-614O4.11 CTRPv2 pan-cancer AAC -0.19 2e-08
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