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PHA-793887

Synonyms

SourcesNames Used
GDSC1000, CTRPv2PHA-793887
PharmacoGx PHA-793887

External IDs

DatabaseIdentifier
Smiles: CC(C)CC(=O)Nc1n[nH]c2c1CN(C(=O)C1CCN(C)CC1)C2(C)C
Pubchem: 46191454

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK7, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to PHA-793887


Feature TypeStandardized
Nominal ANOVA
mRNA YTHDF2 GDSC1000 pan-cancer AAC 0.13 3e-06
mRNA UGT3A2 GDSC1000 pan-cancer AAC 0.16 3e-06
mRNA LEMD3 GDSC1000 pan-cancer AAC 0.14 3e-06
mRNA MFSD5 GDSC1000 pan-cancer AAC -0.13 3e-06
mRNA WISP2 GDSC1000 pan-cancer AAC -0.13 3e-06
mRNA FAM174A GDSC1000 pan-cancer AAC -0.14 3e-06
mRNA SLC35D2 GDSC1000 pan-cancer AAC -0.18 3e-06
mRNA FAM117B GDSC1000 pan-cancer AAC 0.14 3e-06
mRNA HSF2 GDSC1000 pan-cancer AAC 0.14 3e-06
mRNA UEVLD CTRPv2 pan-cancer AAC -0.17 3e-06
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