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PHA-793887

Synonyms

SourcesNames Used
GDSC1000, CTRPv2PHA-793887
PharmacoGx PHA-793887

External IDs

DatabaseIdentifier
Smiles: CC(C)CC(=O)Nc1n[nH]c2c1CN(C(=O)C1CCN(C)CC1)C2(C)C
Pubchem: 46191454

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK7, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to PHA-793887


Feature TypeStandardized
Nominal ANOVA
mRNA FAM76B GDSC1000 pan-cancer AAC 0.17 1e-07
mRNA KRI1 GDSC1000 pan-cancer AAC 0.17 1e-07
mRNA ARHGDIG CTRPv2 pan-cancer AAC 0.17 1e-07
mRNA MBNL2 CTRPv2 pan-cancer AAC -0.18 1e-07
mRNA HS3ST4 GDSC1000 pan-cancer AAC 0.18 1e-07
mRNA THAP9 GDSC1000 pan-cancer AAC 0.16 1e-07
mRNA RPL10A CTRPv2 pan-cancer AAC 0.2 1e-07
mRNA CEP295NL CTRPv2 pan-cancer AAC -0.2 1e-07
mRNA BPTF GDSC1000 pan-cancer AAC 0.16 1e-07
mRNA EVA1A GDSC1000 pan-cancer AAC -0.17 1e-07
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