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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA PRM2 GDSC1000 pan-cancer AAC 0.095 0.004
mRNA VASP GDSC1000 pan-cancer AAC 0.1 0.004
mRNA MBLAC1 GDSC1000 pan-cancer AAC -0.099 0.004
mRNA RBM6 GDSC1000 pan-cancer AAC 0.11 0.004
mRNA GPR162 GDSC1000 pan-cancer AAC 0.11 0.004
mRNA PTS GDSC1000 pan-cancer AAC -0.11 0.004
mRNA DENND1C GDSC1000 pan-cancer AAC 0.13 0.004
mRNA ADRB1 GDSC1000 pan-cancer AAC 0.11 0.004
mRNA IL17RA GDSC1000 pan-cancer AAC 0.1 0.004
mRNA NABP2 GDSC1000 pan-cancer AAC -0.099 0.004
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