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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA CSF1R GDSC1000 pan-cancer AAC 0.37 2e-26
mRNA PTPN7 GDSC1000 pan-cancer AAC 0.32 1e-08
mRNA VSIG4 GDSC1000 pan-cancer AAC 0.32 8e-22
mRNA TRH GDSC1000 pan-cancer AAC 0.31 7e-22
mRNA LST1 GDSC1000 pan-cancer AAC 0.29 2e-12
mRNA FAM78A GDSC1000 pan-cancer AAC 0.27 8e-09
mRNA LYL1 GDSC1000 pan-cancer AAC 0.26 4e-08
mRNA PLPPR3 GDSC1000 pan-cancer AAC 0.26 7e-14
mRNA INPP5D GDSC1000 pan-cancer AAC 0.26 9e-07
mRNA TMC8 GDSC1000 pan-cancer AAC 0.26 6e-08
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