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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA ZBTB14 GDSC1000 pan-cancer AAC -0.1 0.004
mRNA PKM GDSC1000 pan-cancer AAC -0.1 0.004
mRNA GRB2 GDSC1000 pan-cancer AAC 0.11 0.004
mRNA WDFY3 GDSC1000 pan-cancer AAC 0.12 0.003
mRNA SSX2IP GDSC1000 pan-cancer AAC -0.1 0.003
mRNA TMEM185B GDSC1000 pan-cancer AAC -0.11 0.003
mRNA SYNE2 GDSC1000 pan-cancer AAC -0.1 0.003
mRNA CEP170 GDSC1000 pan-cancer AAC 0.11 0.003
mRNA COG4 GDSC1000 pan-cancer AAC -0.099 0.003
mRNA STK10 GDSC1000 pan-cancer AAC 0.13 0.003
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