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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA HIST1H4I GDSC1000 pan-cancer AAC -0.18 3e-06
mRNA RAB11FIP5 CTRPv2 pan-cancer AAC -0.18 2e-05
mRNA ITGB5 CTRPv2 pan-cancer AAC -0.18 2e-05
mRNA ATP6V0E1 CTRPv2 pan-cancer AAC -0.17 2e-05
mRNA MVP CTRPv2 pan-cancer AAC -0.17 9e-06
mRNA PIGT CTRPv2 pan-cancer AAC -0.17 7e-06
mRNA GPX8 CTRPv2 pan-cancer AAC -0.17 0.0001
mRNA B4GALT7 CTRPv2 pan-cancer AAC -0.17 9e-06
mRNA HDLBP CTRPv2 pan-cancer AAC -0.17 1e-05
mRNA FHL2 CTRPv2 pan-cancer AAC -0.17 1e-05
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