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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA ABL2 CTRPv2 pan-cancer AAC -0.13 0.001
mRNA AC002985.3 CTRPv2 pan-cancer AAC -0.14 0.0003
mRNA AC009065.1 CTRPv2 pan-cancer AAC 0.15 5e-05
mRNA AC009336.19 CTRPv2 pan-cancer AAC 0.12 0.002
mRNA AC023908.1 CTRPv2 pan-cancer AAC -0.13 0.002
mRNA AC087350.1 CTRPv2 pan-cancer AAC 0.12 0.003
mRNA AC092835.2 CTRPv2 pan-cancer AAC 0.12 0.0007
mRNA AC096949.1 CTRPv2 pan-cancer AAC 0.14 0.0005
mRNA AC104534.3 CTRPv2 pan-cancer AAC 0.14 0.0002
mRNA ACAP1 CTRPv2 pan-cancer AAC 0.17 0.0007
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