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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA IPP GDSC1000 pan-cancer AAC -0.1 0.004
mRNA DCTN2 GDSC1000 pan-cancer AAC -0.1 0.004
mRNA TMEM106C GDSC1000 pan-cancer AAC -0.1 0.004
mRNA DNAJA2 GDSC1000 pan-cancer AAC 0.1 0.004
mRNA PRKCB GDSC1000 pan-cancer AAC 0.13 0.004
mRNA MFF GDSC1000 pan-cancer AAC -0.1 0.004
mRNA TRIM65 GDSC1000 pan-cancer AAC 0.099 0.004
mRNA ATG16L2 GDSC1000 pan-cancer AAC 0.11 0.004
mRNA MYH10 GDSC1000 pan-cancer AAC -0.11 0.004
mRNA GNPTAB GDSC1000 pan-cancer AAC 0.11 0.004
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