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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA TRIP10 CTRPv2 pan-cancer AAC -0.12 0.003
mRNA ZNF45 CTRPv2 pan-cancer AAC 0.11 0.003
mRNA CCDC27 CTRPv2 pan-cancer AAC 0.11 0.003
mRNA APC2 CTRPv2 pan-cancer AAC 0.15 0.003
mRNA TMEM63C CTRPv2 pan-cancer AAC 0.11 0.003
mRNA GRAMD4 CTRPv2 pan-cancer AAC 0.12 0.003
mRNA PDPK1 GDSC1000 pan-cancer AAC -0.1 0.003
mRNA GAR1 CTRPv2 pan-cancer AAC 0.11 0.003
mRNA KAT6A CTRPv2 pan-cancer AAC 0.11 0.003
mRNA SBDS CTRPv2 pan-cancer AAC -0.12 0.003
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