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ZSTK474

Synonyms

SourcesNames Used
GDSC1000, CTRPv2ZSTK474
PharmacoGx ZSTK474

External IDs

DatabaseIdentifier
Smiles: FC(F)c1nc2ccccc2n1-c1nc(nc(n1)N1CCOCC1)N1CCOCC1
Pubchem: 11647372

Annotated Targets

PIK3CD, PIK3CB, PIK3CG

FDA Approval Status

Not Approved
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Top molecular features associated with response to ZSTK474


Feature TypeStandardized
Nominal ANOVA
mRNA CD53 GDSC1000 pan-cancer AAC 0.33 5e-07
mRNA IKZF1 GDSC1000 pan-cancer AAC 0.29 0.0001
mRNA RCSD1 GDSC1000 pan-cancer AAC 0.29 1e-08
mRNA LRMP GDSC1000 pan-cancer AAC 0.28 9e-09
mRNA NCKAP1L GDSC1000 pan-cancer AAC 0.28 4e-08
mRNA P2RY8 GDSC1000 pan-cancer AAC 0.25 2e-05
mRNA ARHGAP30 CTRPv2 pan-cancer AAC 0.24 4e-05
mRNA ARHGAP45 CTRPv2 pan-cancer AAC 0.23 1e-05
mRNA PIK3CG GDSC1000 pan-cancer AAC 0.23 5e-07
mRNA PTK2B CTRPv2 pan-cancer AAC 0.22 2e-06
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