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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA AC104389.1 CTRPv2 pan-cancer AAC 0.23 8e-11
mRNA AC104389.2 CTRPv2 pan-cancer AAC 0.21 2e-09
mRNA AC138969.4 CTRPv2 pan-cancer AAC 0.19 2e-06
mRNA ACBD3 GDSC1000 pan-cancer AAC -0.091 0.004
mRNA ACRBP GDSC1000 pan-cancer AAC 0.13 0.0002
mRNA ACSBG1 CTRPv2 pan-cancer AAC 0.1 0.004
mRNA ACSL6 CTRPv2 pan-cancer AAC 0.16 1e-05
mRNA ACSM1 CTRPv2 pan-cancer AAC 0.23 1e-10
mRNA ACSM3 CTRPv2 pan-cancer AAC 0.14 7e-05
mRNA ACTN1 GDSC1000 pan-cancer AAC 0.18 2e-05
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