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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA ABL1 GDSC1000 pan-cancer AAC 0.21 3e-10
mRNA ABLIM2 CTRPv2 pan-cancer AAC 0.11 0.002
mRNA AC006538.4 CTRPv2 pan-cancer AAC 0.16 8e-05
mRNA AC010287.1 CTRPv2 pan-cancer AAC 0.1 0.006
mRNA AC015688.3 CTRPv2 pan-cancer AAC 0.14 0.0004
mRNA AC018755.18 CTRPv2 pan-cancer AAC 0.12 0.001
mRNA AC021106.1 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA AC084219.2 CTRPv2 pan-cancer AAC 0.13 0.0006
mRNA AC090154.1 CTRPv2 pan-cancer AAC 0.12 0.003
mRNA AC100821.1 CTRPv2 pan-cancer AAC 0.11 0.002
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