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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA ZNF74 GDSC1000 pan-cancer AAC 0.15 5e-06
mRNA ZNF766 CTRPv2 pan-cancer AAC 0.13 0.001
mRNA ZNF766 GDSC1000 pan-cancer AAC 0.095 0.004
mRNA ZNF77 GDSC1000 pan-cancer AAC 0.12 0.0003
mRNA ZNF776 GDSC1000 pan-cancer AAC 0.095 0.005
mRNA ZNF792 GDSC1000 pan-cancer AAC 0.16 1e-06
mRNA ZNF792 CTRPv2 pan-cancer AAC 0.11 0.005
mRNA ZNF8 CTRPv2 pan-cancer AAC 0.13 0.001
mRNA ZNF804B CTRPv2 pan-cancer AAC 0.16 7e-06
mRNA ZNF823 GDSC1000 pan-cancer AAC 0.099 0.004
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