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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA ZNF776 GDSC1000 pan-cancer AAC 0.095 0.005
mRNA POU4F1 GDSC1000 pan-cancer AAC 0.092 0.005
mRNA GP1BA GDSC1000 pan-cancer AAC 0.088 0.005
mRNA GCNT2 GDSC1000 pan-cancer AAC -0.094 0.005
mRNA STAG3 GDSC1000 pan-cancer AAC -0.094 0.006
mRNA SYNGR3 GDSC1000 pan-cancer AAC -0.089 0.006
mRNA BICD2 CTRPv2 pan-cancer AAC -0.11 0.006
mRNA AACS GDSC1000 pan-cancer AAC -0.09 0.006
mRNA SLC9A8 GDSC1000 pan-cancer AAC -0.095 0.006
mRNA CFD GDSC1000 pan-cancer AAC 0.091 0.006
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