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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA GIMAP6 GDSC1000 pan-cancer AAC 0.22 7e-11
mRNA AC104389.1 CTRPv2 pan-cancer AAC 0.23 8e-11
mRNA LAIR2 CTRPv2 pan-cancer AAC 0.24 9e-11
mRNA HBB CTRPv2 pan-cancer AAC 0.23 9e-11
mRNA SPTA1 CTRPv2 pan-cancer AAC 0.23 1e-10
mRNA ACSM1 CTRPv2 pan-cancer AAC 0.23 1e-10
mRNA GAB3 GDSC1000 pan-cancer AAC 0.25 1e-10
mRNA TUBB1 GDSC1000 pan-cancer AAC 0.2 2e-10
mRNA HBG1 CTRPv2 pan-cancer AAC 0.22 2e-10
mRNA HBG2 CTRPv2 pan-cancer AAC 0.22 2e-10
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