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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA TCEA1 GDSC1000 pan-cancer AAC 0.093 0.005
mRNA MID1 GDSC1000 pan-cancer AAC -0.11 0.005
mRNA ANKRD63 CTRPv2 pan-cancer AAC 0.11 0.005
mRNA DLG4 GDSC1000 pan-cancer AAC 0.096 0.005
mRNA MAPK8IP2 CTRPv2 pan-cancer AAC 0.11 0.005
mRNA ZNF706 GDSC1000 pan-cancer AAC 0.09 0.005
mRNA ATP6V0A4 CTRPv2 pan-cancer AAC 0.1 0.005
mRNA C7orf72 GDSC1000 pan-cancer AAC -0.092 0.005
mRNA HLA-DRA GDSC1000 pan-cancer AAC -0.11 0.005
mRNA SELT GDSC1000 pan-cancer AAC -0.087 0.005
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